The first report of 1′-homo-N-1,2,3-triazol-bicyclic carbonucleosides (7a and 7b) is described herein. Azide-enolate (3+2) cycloaddition afforded the synthesis of this novel type of compound. Antifungal activity was evaluated ...

A small library of diverse 1,1-diaryl-2-(1,2,3)triazol-1-yl-ethanol derivatives was designed and prepared from CuAAC reaction as the key step. The molecular structure of some representative compounds was unambiguously ...